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VRT752271

A ERK1/ERK2 inhibitor
Catalog #: B1679
SKU-Size Size Price Qty
B1679-5 5 mg
$115.00
B1679-25 25 mg
$440.00
More Sizes Get Quote

Product Details

Alternate Name VRT752271; Ulixertinib; VRT752271; VRT-752271; BVD-523; BVD523; BVD 523; N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-[5-chloro-2-(propan-2-ylamino)pyridin-4-yl]-1H-pyrrole-2-carboxamide
Appearance Solid
CAS # 869886-67-9
Molecular Formula C₂₁H₂₂Cl₂N₄O₂
Molecular Weight 433.33
Purity >98%
Solubility DMSO
SMILES CC(C)NC1=NC=C(C(=C1)C2=CNC(=C2)C(=O)NC(CO)C3=CC(=CC=C3)Cl)Cl
InChi InChI=1S/C21H22Cl2N4O2/c1-12(2)26-20-8-16(17(23)10-25-20)14-7-18(24-9-14)21(29)27-19(11-28)13-4-3-5-15(22)6-13/h3-10,12,19,24,28H,11H2,1-2H3,(H,25,26)(H,27,29)/t19-/m1/s1
InChi Key KSERXGMCDHOLSS-LJQANCHMSA-N
PubChem CID 11719003
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

VRT752271 is a reversible, ATP-competitive inhibitor of ERK1 and ERK2 kinases, with IC50 of <0.3 nM against ERK2.


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