Call 408.493.1800 | Fax 408.493.1801 | Toll Free 800.891.9699 (US Only) | Email: [email protected]


A potent G9a inhibitor
Catalog #: 2605
SKU-Size Size Price Qty
2605-5 5 mg
2605-25 25 mg
More Sizes Get Quote

Product Details

Alternate Name [N-(1-(cyclohexylmethyl)piperidin-4-yl)-2-(4-isopropyl-1,4-diazepan-1-yl)-6-methoxy-7-(3-(piperidin-1-yl)propoxy)quinazolin-4-amine
Appearance White to off-white solid
CAS # 1320288-19-4
Molecular Formula C₃₇H₆₁N₇O₂
Molecular Weight 635.93
Purity >98% by HPLC
Solubility DMSO (~30 mg/ml)
InChi InChI=1S/C35H59N7O2/c1-6-39(4)16-11-23-44-33-25-31-30(24-32(33)43-5)34(38-35(37-31)42-18-10-17-41(21-22-42)27(2)3)36-29-14-19-40(20-15-29)26-28-12-8-7-9-13-28/h24-25,27-29H,6-23,26H2,1-5H3,(H,36,37,38)
Handling Protect from air and light
Storage Conditions -20 ̊C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.


UNC0631 is a potent and selective inhibitor of G9a activity in vitro (IC₅₀ = 4 nM) and G9a/GLP-mediated dimethylation of histone 3 on lysine 9 in MDA-MB-231 cells (IC₅₀ = 25 nM). It potently inhibits G9a/GLP activity in a variety of cancer cell lines as well as in the human fetal lung IMR-90 cell line. Also displays excellent separation of functional potency versus cell toxicity.

Why buy BioVision Products?
Global Presence
Technical Support
BioVision aims to provide our customers innovative tools for accelerating drug discovery and biological research. BioVision offers >8,000 products including the most comprehensive array of assay kits for key targets in Metabolic pathways.
BioVision is committed to providing the highest quality products at a competitive price.
We have a broad network of global distributors who are ready to address your research needs and ensure fast delivery.
Our highly trained Technical Support team provides comprehensive product support and is dedicated to resolving your issues quickly and efficiently.