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TC-E 5002

An inhibitor of KDM2/7
Catalog #: B2856
SKU-Size Size Price Qty
B2856-1 1 mg
B2856-5 5 mg
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Product Details

Alternate Name 3-[9-cyclopropylnonanoyl(hydroxy)amino]propanoic acid; N-(9-Cyclopropyl-1-oxononyl)-N-hydroxy-beta-alanine; 3-(9-cyclopropyl-N-hydroxynonanamido)propanoic acid
Appearance A crystalline solid
CAS # 1453071-47-0
Molecular Formula C₁₅H₂₇NO₄
Molecular Weight 285.38
Purity ≥98%
Solubility ~30 mg/ml in DMSO
~50 mg/ml in Ethanol
~10 mg/ml in DMF
~0.25 mg/ml in PBS, pH 7.2
InChi InChI=1S/C15H27NO4/c17-14(16(20)12-11-15(18)19)8-6-4-2-1-3-5-7-13-9-10-13/h13,20H,1-12H2,(H,18,19)
PubChem CID 71735843
Handling Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
Storage Conditions -20ºC
Shipping Conditions RT
USAGE For Research Use Only! Not For Use in Humans.


TC-E 5002 is an inhibitor of the histone lysine demethylase (KDM) subfamily KDM2/7. It potently inhibits KDM2A, KDM7A and KDM7B with an IC₅₀ of 6.8 μM, 0.2 μM and 1.2 μM respectively. It inhibits the growth of KYSE150 and HeLa cells with GI₅₀ values of 16 µM and 40 µM respectively and arrests cells in the G0/G1 phase of the cell cycle. It inhibits demethylation of H3K27me2 at similar concentrations.

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