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PKI-402

A reversible and potent dual inhibitor of PI3K/mTOR
Catalog #: B1715

In stock

SKU-Size Size Price Qty
B1715-1 1 mg
$125.00
B1715-5 5 mg
$495.00

Product Details

Alternate Name PKI-402; PKI 402; PKI402; 1-[4-(3-ethyl-7-morpholin-4-yltriazolo[4,5-d]pyrimidin-5-yl)phenyl]-3-[4-(4-methylpiperazine-1-carbonyl)phenyl]urea
Appearance Solid
CAS # 173204-81-3
Molecular Formula C₂₉H₃₄N₁₀O₃
Molecular Weight 570.65
Purity >98%
Solubility DMSO
SMILES CCN1C2=C(C(=NC(=N2)C3=CC=C(C=C3)NC(=O)NC4=CC=C(C=C4)C(=O)N5CCN(CC5)C)N6CCOCC6)N=N1
InChi InChI=1S/C29H34N10O3/c1-3-39-27-24(34-35-39)26(37-16-18-42-19-17-37)32-25(33-27)20-4-8-22(9-5-20)30-29(41)31-23-10-6-21(7-11-23)28(40)38-14-12-36(2)13-15-38/h4-11H,3,12-19H2,1-2H3,(H2,30,31,41)
InChi Key ZAXFYGBKZSQBIV-UHFFFAOYSA-N
PubChem CID 44187953
MDL Number MFCD18251484
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

PKI-402 is a reversible, potent dual inhibitor of PI3K/mTOR with IC50 values of 2 nM/7 nM/16 nM/14 nM and 3 nM for PI3Kα/β/γ/δ and mTOR, respectively.


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