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PIK75

Inhibitor of PI3K isoform p110α
Catalog #: B1668

In stock

SKU-Size Size Price Qty
B1668-5 5 mg
$60.00
B1668-25 25 mg
$195.00

Product Details

Alternate Name PIK75 , PIK75; PIK 75; PIK-75 Hydrochloride; PIK75 Hydrochloride; PIK 75 Hydrochloride; (E)-N'-((6-bromoH-imidazo[1,2-a]pyridin-3-yl)methylene)-N,2-dimethyl-5-nitrobenzenesulfonohydrazide hydrochloride; PIK-75 Hydrochloride; PIK75 Hydrochloride; PIK 75 Hydrochloride
Appearance Solid
CAS # 372196-77-5
Molecular Formula C₁₆H₁₅BrClN₅O₄S
Molecular Weight 488.74
Purity >98%
Solubility DMSO
SMILES CC1=C(C=C(C=C1)[N+](=O)[O-])S(=O)(=O)N(C)N=CC2=CN=C3N2C=C(C=C3)Br.Cl
InChi InChI=1S/C16H14BrN5O4S.ClH/c1-11-3-5-13(22(23)24)7-15(11)27(25,26)20(2)19-9-14-8-18-16-6-4-12(17)10-21(14)16;/h3-10H,1-2H3;1H/b19-9+;
InChi Key VOUDEIAYNKZQKM-MYHMWQFYSA-N
PubChem CID 45265864
MDL Number MFCD12546130
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

PIK-75 is a p110α inhibitor with IC50 of 5.8 nM (200-fold more potently than p110β), isoform-specific mutants at Ser773, and also potently inhibits DNA-PK with IC50 of 2 nM.


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