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K252a

A selective protein kinase inhibitor
Catalog #: 2013
SKU-Size Size Price Qty
2013-500 500 µg
$90.00
2013-1000 1 mg
$140.00
More Sizes Get Quote

Product Details

Alternate Name SF 2370
Appearance White solid
CAS # 99533-80-9
Molecular Formula C₂₇H₂₁N₃O₅
Molecular Weight 467.47
Purity ≥98% by HPLC
Solubility DMSO (100 mg/ml)
SMILES CC12C(CC(O1)N3C4=CC=CC=C4C5=C6C(=C7C8=CC=CC=C8N2C7=C53)CNC6=O)(C(=O)OC)O
InChi InChI=1S/C27H21N3O5/c1-26-27(33,25(32)34-2)11-18(35-26)29-16-9-5-3-7-13(16)20-21-15(12-28-24(21)31)19-14-8-4-6-10-17(14)30(26)23(19)22(20)29/h3-10,18,33H,11-12H2,1-2H3,(H,28,31)/t18-,26+,27?/m1/s1
InChi Key KOZFSFOOLUUIGY-UHOLRESSSA-N
PubChem CID 127357
MDL Number MFCD00161522
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

An analog of Staurosporine (Cat. No. 1048) that acts as a non-selective protein kinase inhibitor. Iinhibits PKA (Ki = 18 nM), PKC (Ki = 25 nM), and PKG (Ki = 20 nM). Potently inhibits CaMK (Ki = 1.8 nM), competitively with ATP and noncompetitively with the substrate.


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