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A potent bromodomain inhibitor
Catalog #: 2628
SKU-Size Size Price Qty
2628-1 1 mg
2628-5 5 mg
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Product Details

Alternate Name (4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide; GSK525762
Appearance Off-white solid
CAS # 1260907-17-2
Molecular Formula C₂₂H₂₂ClN₅O₂
Molecular Weight 423.9
Purity >98% by HPLC
Solubility DMSO or EtOH
InChi nChI=1S/C22H22ClN5O2/c1-4-24-20(29)12-18-22-27-26-13(2)28(22)19-10-9-16(30-3)11-17(19)21(25-18)14-5-7-15(23)8-6-14/h5-11,18H,4,12H2,1-3H3,(H,24,29)/t18-/m0/s1
PubChem CID 46943432
Handling Protect from air and light
Storage Conditions -20 ̊C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.


I-BET762 (GSK525762) is a highly potent, selective and cell-permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 (IC₅₀ of ~35 nM). It inhibits myeloma cell proliferation and suppresses the production of proinflammatory proteins by macrophages and blocks acute inflammation.

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