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GSK-961081

A bi-functional molecule with both muscarinic antagonism and β2-agonism (MABA) properties.
Catalog #: B1590

In stock

SKU-Size Size Price Qty
B1590-5 5 mg
$175.00
B1590-25 25 mg
$695.00

Product Details

Alternate Name  (R)-1-(3-((2-chloro-4-(((2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroquinolin-5-yl)ethyl)amino)methyl)-5-methoxyphenyl)amino)-3-oxopropyl)piperidin-4-yl [1,1'-biphenyl]-2-ylcarbamate; Batefenterol;TD-5959
Appearance Crystalline solid
CAS # 743461-65-6 
Molecular Formula C₄₀H₄₂ClN₅O₇ 
Molecular Weight 740.25
Purity ≥98% by HPLC
Solubility DMSO
SMILES COC1=CC(=C(C=C1CNCC(C2=C3C=CC(=O)NC3=C(C=C2)O)O)Cl)NC(=O)CCN4CCC(CC4)OC(=O)NC5=CC=CC=C5C6=CC=CC=C6
InChi InChI=1S/C40H42ClN5O7/c1-52-36-22-33(31(41)21-26(36)23-42-24-35(48)29-11-13-34(47)39-30(29)12-14-37(49)45-39)43-38(50)17-20-46-18-15-27(16-19-46)53-40(51)44-32-10-6-5-9-28(32)25-7-3-2-4-8-25/h2-14,21-22,27,35,42,47-48H,15-20,23-24H2,1H3,(H,43,50)(H,44,51)(H,45,49)/t35-/m0/s1
InChi Key URWYQGVSPQJGGB-DHUJRADRSA-N
PubChem CID 10372836
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

GSK-961081 is a bi-functional molecule with both muscarinic antagonism and β2-agonism (MABA) properties. GSK-961081 displays high affinity for hM2 (Ki = 1.4 nM), hM3 muscarinic receptors (Ki = 1.3 nM) and hβ2-adrenoceptors (Ki = 3.7 nM). 


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