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GSK-3787

A potent PPARδ antagonist
Catalog #: 2400
SKU-Size Size Price Qty
2400-5 5 mg
$95.00
2400-25 25 mg
$375.00
More Sizes Get Quote

Product Details

Alternate Name 4-Chloro-N-(2-{[5-(trifluoromethyl)-2-pyridyl]sulfonyl}ethyl)benzamide
Appearance White solid
CAS # 188591-46-0
Molecular Formula C₁₅H₁₂ClF₃N₂O₃S
Molecular Weight 392.78
Purity ≥98% by TLC
Solubility DMSO (~30 mg/ml)
SMILES C1=CC(=CC=C1C(=O)NCCS(=O)(=O)C2=NC=C(C=C2)C(F)(F)F)Cl
InChi InChI=1S/C15H12ClF3N2O3S/c16-12-4-1-10(2-5-12)14(22)20-7-8-25(23,24)13-6-3-11(9-21-13)15(17,18)19/h1-6,9H,7-8H2,(H,20,22)
InChi Key JFUIMTGOQCQTPF-UHFFFAOYSA-N
PubChem CID 2800647
MDL Number MFCD00099612
Handling Protect from light and air
Storage Conditions -20 ̊C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

GSK-3787 is a selective and irreversible antagonist of the peroxisome proliferator-activated receptor delta (PPARδ) (plC₅₀ = 6.6). It covalently binds to Cys 249 in the PPARδ binding site.


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