Call 408.493.1800 | Fax 408.493.1801 | Toll Free 800.891.9699 (US Only) | Email: [email protected]

GSK-121 trifluoroacetate

A novel protein arginine deiminase 4 (PAD4) inhibitor
Catalog #: B1034
SKU-Size Size Price Qty
B1034-500 500 µg
$75.00
B1034-1000 1 mg
$125.00
More Sizes Get Quote

Product Details

Alternate Name (3-​amino-1-​piperidinyl)​[1-​methyl-​2-​(1-​methyl-​1H-​indol-​2-​yl)​-​1H-​benzimidazol-​5-​yl]​-methanone, 2,​2,​2-​trifluoroacetate
Appearance Crystalline solid
CAS # 1652591-80-4
Molecular Formula C₂₃H₂₅N₅O •CF₃COOH
Molecular Weight 501.5
Purity ≥98%
Solubility DMSO (~30 mg/ml)
SMILES O=C(N1CC(N)CCC1)C2=CC=C3N(C)C(C(N4C)=CC5=C4C=CC=C5)=NC3=C2.OC(C(F)(F)F)=O
InChi InChI=1S/C23H25N5O.C2HF3O2/c1-26-19-8-4-3-6-15(19)13-21(26)22-25-18-12-16(9-10-20(18)27(22)2)23(29)28-11-5-7-17(24)14-28;3-2(4,5)1(6)7/h3-4,6,8-10,12-13,17H,5,7,11,14,24H2,1-2H3;(H,6,7)
InChi Key CUCLWQZRCAQPJM-UHFFFAOYSA-N
Handling Protect from air and moisture
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

GSK-121 is a novel protein arginine deiminase 4 (PAD4) inhibitor. GSK-121 was shown to inhibit the citrullination of PAD4 target proteins in a functional assay with an IC₅₀ value of 3.2 µM.


Why buy BioVision Products?
Innovation
Affordability
Global Presence
Technical Support
BioVision aims to provide our customers innovative tools for accelerating drug discovery and biological research. BioVision offers >8,000 products including the most comprehensive array of assay kits for key targets in Metabolic pathways.
BioVision is committed to providing the highest quality products at a competitive price.
We have a broad network of global distributors who are ready to address your research needs and ensure fast delivery.
Our highly trained Technical Support team provides comprehensive product support and is dedicated to resolving your issues quickly and efficiently.