GDC-0941 Dimethanesulfonate

A potent, selective, inhibitor of pan-class I PI3 kinase
Catalog #: 9618 | abID:

Product Details

Alternate Name 4-[2-(1H-indazol-4-yl)-6-[(4-methylsulfonylpiperazin-1-yl)methyl]thieno[3,2-d]pyrimidin-4-yl]morpholine;methanesulfonic acid; Pictilisib
Appearance White to off-white solid
CAS # 957054-33-0
Molecular Formula C₂₅H₃₅N₇O₉S₄
Molecular Weight 705.85
Purity ≥98% by HPLC
Solubility DMSO (>10 mg/ml)
InChi InChI=1S/C23H27N7O3S2.2CH4O3S/c1-35(31,32)30-7-5-28(6-8-30)15-16-13-20-21(34-16)23(29-9-11-33-12-10-29)26-22(25-20)17-3-2-4-19-18(17)14-24-27-19;2*1-5(2,3)4/h2-4,13-14H,5-12,15H2,1H3,(H,24,27);2*1H3,(H,2,3,4)
PubChem CID 56972143
Handling Protect from air and moisture
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.


GDC-0941 is a potent, selective, inhibitor of pan-class I PI3 kinase (PI3K), with IC₅₀ values of 3, 33, 3, 75, 1230 and 580 nM for p110 α, β, δ and γ isoforms, DNA-PK and mTOR respectively. Displays antineoplastic activity.

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Yichun Zhu. Interferon gamma induces inflammatory responses through the interaction of CEACAM1 and PI3K in airway epithelial cells. J Transl Med May-19. 31072323.
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