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XMD17-109

A ERK-5 inhibitor
Catalog #: B1685

In stock

SKU-Size Size Price Qty
B1685-5 5 mg
$175.00
B1685-25 25 mg
$690.00
More Sizes Get Quote

Product Details

Alternate Name XMD17-109; XMD17 109; XMD17109; 11-cyclopentyl-2-[2-ethoxy-4-[4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]anilino]-5-methylpyrimido[4,5-b][1,4]benzodiazepin-6-one
Appearance Solid
CAS # 1435488-37-1
Molecular Formula C₃₆H₄₆N₈O₃
Molecular Weight 638.8
Purity >98%
Solubility DMSO
SMILES CCOC1=C(C=CC(=C1)C(=O)N2CCC(CC2)N3CCN(CC3)C)NC4=NC=C5C(=N4)N(C6=CC=CC=C6C(=O)N5C)C7CCCC7
InChi InChI=1S/C36H46N8O3/c1-4-47-32-23-25(34(45)43-17-15-26(16-18-43)42-21-19-40(2)20-22-42)13-14-29(32)38-36-37-24-31-33(39-36)44(27-9-5-6-10-27)30-12-8-7-11-28(30)35(46)41(31)3/h7-8,11-14,23-24,26-27H,4-6,9-10,15-22H2,1-3H3,(H,37,38,39)
InChi Key XVBGRTMNFNMINE-UHFFFAOYSA-N
PubChem CID 71604307
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

XMD17-109 is a novel, specific ERK-5 inhibitor, which inhibits the ERK5-mediated AP1 transcriptional activity at 30 μM, and has an EC50 of 4.2 μM.


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