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A potent, and selective BET (bromodomain and extra terminal family of proteins) inhibitor
Catalog #: B1201
SKU-Size Size Price Qty
B1201-5 5 mg
B1201-25 25 mg
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Product Details

Alternate Name (S)-2-(6-(4-chlorophenyl)-1-methyl-4H-benzo[c]isoxazolo[4,5-e]azepin-4-yl)acetamide
Appearance White Solid
CAS # 1380087-89-7 
Molecular Formula C₂₀H₁₆ClN₃O₂
Molecular Weight 365.82
Purity ≥98% by HPLC
Solubility DMSO(>3 mg/ml)
InChi InChI=1S/C20H16ClN3O2/c1-11-18-14-4-2-3-5-15(14)19(12-6-8-13(21)9-7-12)23-16(10-17(22)25)20(18)26-24-11/h2-9,16H,10H2,1H3,(H2,22,25)
PubChem CID 76534645
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.


CPI-0610 is a potent, selective BET (bromodomain and extra terminal family of proteins) inhibitor and inhibits BRD4-BD1 with IC₅₀ of 39 nM. It potentially demonstrates anti-neoplastic activity by binding acetylated lysine recognition motifs on the bromodomain of BET proteins, thus preventing the interaction of BET proteins and acetylated histone peptides.

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