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CCT-251921

A potent, selective, and orally bioavailable CDK8 inhibitor
Catalog #: B2502
SKU-Size Size Price Qty
B2502-1 1 mg
$85.00
B2502-5 5 mg
$335.00
More Sizes Get Quote

Product Details

Alternate Name 8-(2-amino-3-chloro-5-(1-methyl-1H-indazol-5-yl)pyridin-4-yl)-2,8-diazaspiro[4.5]decan-1-one; CCT251921; CCT 251921
Appearance Crystalline solid
CAS # 1607837-31-9
Molecular Formula C₂₁H₂₃ClN₆O
Molecular Weight 410.90
Purity ≥98% by HPLC
Solubility >25 mg/ml in DMSO
SMILES CN1C2=C(C=C(C=C2)C3=CN=C(C(=C3N4CCC5(CCNC5=O)CC4)Cl)N)C=N1
InChi InChI=1S/C21H23ClN6O/c1-27-16-3-2-13(10-14(16)11-26-27)15-12-25-19(23)17(22)18(15)28-8-5-21(6-9-28)4-7-24-20(21)29/h2-3,10-12H,4-9H2,1H3,(H2,23,25)(H,24,29)
InChi Key VPJXPDLMACOGIZ-UHFFFAOYSA-N
PubChem CID 74222277
Handling Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
Storage Conditions -20ºC
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

CCT-251921 is a potent, selective, small-molecule modulator of the mediator complex-associated kinases CDK8 and CDK19 (IC₅₀, CDK8 = 2.3 nM; CDK19 = 2.6 nM).


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