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BIIE 0246

Potent, selective non-peptide NPY Y2 receptor antagonist
Catalog #: B2424

In stock

SKU-Size Size Price Qty
B2424-1 1 mg
$155.00
B2424-5 5 mg
$595.00
More Sizes Get Quote

Product Details

Alternate Name N-[(1S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1 -[2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide
Appearance White solid
CAS # 246146-55-4
Molecular Formula C₄₉H₅₇N₁₁O₆
Molecular Weight 896.06
Purity ≥98% by HPLC
Solubility >50 mg/ml in DMSO
SMILES C1CCC(C1)(CC(=O)NC(CCCN=C(N)N)C(=O)NCCN2C(=O)N(N(C2=O)C3=CC=CC=C3)C4=CC=CC=C4)CC(=O) N5CCN (CC5)C6C7=CC=CC=C7C(=O)NC8=CC=CC=C68
InChi InChI=1S/C49H57N11O6/c50-46(51)53-25-13-22-40(45(64)52-26-27-58-47(65)59(34-14-3-1-4-15-34)60(48(58) 66)35-16-5-2-6-17-35)54-41(61)32-49(23-11-12-24-49)33-42(62)56-28-30-57(31-29-56)43-36-18-7-8-19-37(36) 44(63)55-39-21-10-9-20-38(39)43/h1-10,14-21,40,43H,11-13,22-33H2,(H,52,64)(H,54,61)(H,55,63)(H4,50,51,53)/t40-,43?/m0/s1
InChi Key RSJAXPUYVJKAAA-JPGJPTAESA-N
PubChem CID 9811493
Handling Do not take internally. Wear gloves and mask when handling the product! Avoid contact by all modes of exposure.
Storage Conditions -20ºC
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.

Details

BIIE 0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor (IC₅₀ = 15 nM). BIIE 0246 displays > 650-fold selectivity over Y1, Y4 and Y5 receptors.


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