Call 408.493.1800 | Fax 408.493.1801 | Toll Free 800.891.9699 (US Only) | Email: [email protected]

BAG 956

A dual PI3K/PDK-1 inhibitor
Catalog #: 2456
SKU-Size Size Price Qty
2456-5 5 mg
2456-25 25 mg
More Sizes Get Quote

Product Details

Alternate Name α,α,-Dimethyl-4-[2-methyl-8-[2-(3-pyr​idinyl)ethynyl]-1H-imidazo[4,5-c]quinolin-1-yl]-be​nzeneacetonitrile
Appearance Red solid
CAS # 853910-02-8
Molecular Formula C₂₈H₂₁N₅
Molecular Weight 427.5
Purity ≥98% by HPLC
Solubility DMSO (~15 mg/ml) or EtOH (~7 mg/ml)
InChi InChI=1S/C28H21N5/c1-19-32-26-17-31-25-13-8-20(6-7-21-5-4-14-30-16-21)15-24(25)27(26)33(19)23-11-9-22(10-12-23)28(2,3)18-29/h4-5,8-17H,1-3H3
PubChem CID 24882589
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.


A potent, ATP-competitive, dual PI3K/PDK-1 inhibitor in vitro and in vivo (IC₅₀ = 56, 444, 34, 117 and 240 nM for PI3K p110-α ,β,d, γ, and PDK1 kinases, respectively). Displays anticancer properties.

Why buy BioVision Products?
Global Presence
Technical Support
BioVision aims to provide our customers innovative tools for accelerating drug discovery and biological research. BioVision offers >8,000 products including the most comprehensive array of assay kits for key targets in Metabolic pathways.
BioVision is committed to providing the highest quality products at a competitive price.
We have a broad network of global distributors who are ready to address your research needs and ensure fast delivery.
Our highly trained Technical Support team provides comprehensive product support and is dedicated to resolving your issues quickly and efficiently.