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BAY-876

A highly selective GLUT1 inhibitor
SKU: B1572

Availability: In stock

SKU-Size Size Price Qty
B1572-5 5 mg
$175.00
B1572-25 25 mg
$695.00

Details

BAY-876 is a highly selective GLUT1 inhibitor (IC₅₀ = 2 mM). Displays good metabolic stability in vitro and high oral bioavailability in vivo.

Product Details

Alternate Name N4-[1-[(4-cyanophenyl)methyl]-5-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]-7-fluoro-2,4-Quinolinedicarboxamide
Appearance Crystalline solid
CAS # 1799753-84-6
Molecular Formula C₂₄H₁₆F₄N₆O₂
Molecular Weight 496.42
Purity ≥98% by HPLC
Solubility DMSO
SMILES CC1=C(C(=NN1CC2=CC=C(C=C2)C#N)C(F)(F)F)NC(=O)C3=CC(=NC4=C3C=CC(=C4)F)C(=O)N
InChi InChI=1S/C24H16F4N6O2/c1-12-20(21(24(26,27)28)33-34(12)11-14-4-2-13(10-29)3-5-14)32-23(36)17-9-19(22(30)35)31-18-8-15(25)6-7-16(17)18/h2-9H,11H2,1H3,(H2,30,35)(H,32,36)
InChi Key BKLJDIJJOOQUFG-UHFFFAOYSA-N
PubChem CID 118191391
Handling Protect from air and light
Storage Conditions -20°C
Shipping Conditions Gel Pack
USAGE For Research Use Only! Not For Use in Humans.
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